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dc.contributor.author
Fernandez, Ariel
dc.date.available
2023-09-19T10:04:41Z
dc.date.issued
2021-07
dc.identifier.citation
Fernandez, Ariel; Artificial Intelligence Deconstructs Drug Targeting in Vivo by Leveraging a Transformer Platform; American Chemical Society; ACS Medicinal Chemistry Letters; 12; 7; 7-2021; 1052-1055
dc.identifier.issn
1948-5875
dc.identifier.uri
http://hdl.handle.net/11336/211913
dc.description.abstract
Lead optimization in structure-based drug design ultimately requires that the therapeutic agent be evaluated in the cellular context. However, the in vivo control of the target structure remains unyielding to computational modeling. This situation may change as transformer technologies enable a deconstruction of in vivo cooperativity steering drug-induced protein folding.
dc.format
application/pdf
dc.language.iso
eng
dc.publisher
American Chemical Society
dc.rights
info:eu-repo/semantics/restrictedAccess
dc.rights.uri
https://creativecommons.org/licenses/by-nc-sa/2.5/ar/
dc.subject
ARTIFICIAL INTELLIGENCE
dc.subject
DRUG-INDUCED PROTEIN FOLDING
dc.subject
IN VIVO PROTEIN FOLDING
dc.subject
MOLECULAR DYNAMICS
dc.subject
STRUCTURE-BASED DRUG DESIGN
dc.subject
TRANSFORMER
dc.subject.classification
Ciencias de la Información y Bioinformática
dc.subject.classification
Ciencias de la Computación e Información
dc.subject.classification
CIENCIAS NATURALES Y EXACTAS
dc.title
Artificial Intelligence Deconstructs Drug Targeting in Vivo by Leveraging a Transformer Platform
dc.type
info:eu-repo/semantics/article
dc.type
info:ar-repo/semantics/artículo
dc.type
info:eu-repo/semantics/publishedVersion
dc.date.updated
2023-09-14T17:39:40Z
dc.journal.volume
12
dc.journal.number
7
dc.journal.pagination
1052-1055
dc.journal.pais
Estados Unidos
dc.description.fil
Fil: Fernandez, Ariel. Consejo Nacional de Investigaciones Científicas y Técnicas. Centro Científico Tecnológico Conicet - Bahía Blanca. Instituto de Química del Sur. Universidad Nacional del Sur. Departamento de Química. Instituto de Química del Sur; Argentina
dc.journal.title
ACS Medicinal Chemistry Letters
dc.relation.alternativeid
info:eu-repo/semantics/altIdentifier/doi/http://dx.doi.org/10.1021/acsmedchemlett.1c00237
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